Title of article
(4-Substituted-phenyl)-(5H-10,11-dihydro-pyrrolo [2,1-c][1,4] benzodiazepin-10-yl)-methanone derivatives as vasopressin receptor modulators
Author/Authors
Aranapakam M. Venkatesan، نويسنده , , George T. Grosu، نويسنده , , Amedeo A. Failli، نويسنده , , Peter S. Chan، نويسنده , , Joseph Coupet، نويسنده , , Trina Saunders، نويسنده , , Hussain Mazandarani، نويسنده , , Xun Ru، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 2005
Pages
4
From page
5003
To page
5006
Abstract
Synthesis and structure–activity relationships (SAR) of arginine vasopressin (AVP) receptor modulators are described. Potent and selective compounds are prepared when the amide linkage connecting rings A and B of VPA-985 is replaced with a bond, C O, –O–, –S–, or –SO2– bond.
Keywords
Vasopressin receptor modulators
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
2005
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
796118
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