• Title of article

    Toll-like receptor 2 antagonists. Part 1: Preliminary SAR investigation of novel synthetic phospholipids

  • Author/Authors

    Mark R. Spyvee، نويسنده , , Huiming Zhang، نويسنده , , Lynn D. Hawkins، نويسنده , , Jesse C. Chow، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2005
  • Pages
    5
  • From page
    5494
  • To page
    5498
  • Abstract
    Novel synthetic phospholipid compound 1 was discovered to be an antagonist of human toll-like receptor 2 (TLR2) signaling. In a preliminary SAR campaign we synthesized several analogues of 1 and found that considerable structural changes could be made without loss of TLR2 antagonistic activity.
  • Keywords
    TLR2 , TLR2 antagonist , Synthetic phospholipid , Toll-like receptor
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2005
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    796215