• Title of article

    Synthesis and biological evaluation of simplified mycothiazole analogues

  • Author/Authors

    Graciela Mahler، نويسنده , , Gloria Serra، نويسنده , , Sylvia Dematteis، نويسنده , , Jenny Salda?a، نويسنده , , Laura Dom?nguez، نويسنده , , Eduardo Manta، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2006
  • Pages
    3
  • From page
    1309
  • To page
    1311
  • Abstract
    Thiazoline and oxazoline analogues of the natural product mycothiazole were synthesized from a common intermediate and evaluated in vitro against HCT-15 colon cancer cells and L4 larvae of nematode Nippostrongylus brasiliensis. The nature of the heterocyclic moiety seems to modulate the cytotoxic or anthelmintic activity.
  • Keywords
    Mycothiazole , Oxazolines , anthelmintic , HTC-15 colon cells , Thiazolines , Deoxo-Fluor
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2006
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    796566