• Title of article

    Design and synthesis of novel 5,6-disubstituted uracil derivatives as potent inhibitors of thymidine phosphorylase

  • Author/Authors

    Radim Nencka، نويسنده , , Ivan Votruba، نويسنده , , Hubert H?ebabeck?، نويسنده , , Eva Tlou?t’ov?، نويسنده , , Kv?ta Horsk?، نويسنده , , Milena Masoj?dkov?، نويسنده , , Anton?n Hol?، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2006
  • Pages
    3
  • From page
    1335
  • To page
    1337
  • Abstract
    We report on a series of novel 5,6-disubstituted uracils with significant inhibitory activity against human and Escherichia coli thymidine phosphorylases. Bis-uracil conjugates were identified as the most potent inhibitors of TPs in this study.
  • Keywords
    Thymidine phosphorylase inhibitor , Disubstituted uracils , angiogenesis
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2006
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    796572