• Title of article

    Synthesis and antitumor activity of icogenin and its analogue

  • Author/Authors

    Shujie Hou، نويسنده , , Peng Xu، نويسنده , , Jiong-liang Zhou، نويسنده , , Dequan Yu، نويسنده , , Pingsheng Lei، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2006
  • Pages
    5
  • From page
    2454
  • To page
    2458
  • Abstract
    Natural saponin icogenin, namely 25(S)-22-O-methyl-furost-5-en-3β,26-dio-3-O-α-l-rhamnopyranosyl-(1 → 2)-[β-d-glucopyranosyl-(1 → 3)]-β-d-glucopyranoside, and one of its analogues, 25(S)-22-O-methyl-furost-5-en-3β,26-dio-3-O-α-l-rhamnopyranosyl-(1 → 2)-[β-d-glucopyranosyl-(1 → 3)]-α-d-glucopyranoside, were first synthesized via line strategy and convergent approach, respectively. It was observed that icogenin and its analogue show potent antitumor activity in vitro.
  • Keywords
    Saponin , Icogenin , Glycosylation , cytotoxicity
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2006
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    796800