• Title of article

    Synthesis and evaluation of a mechanism-based inhibitor of a 3-deoxy-d-arabino heptulosonate 7-phosphate synthase

  • Author/Authors

    Scott R. Walker، نويسنده , , Emily J. Parker، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2006
  • Pages
    4
  • From page
    2951
  • To page
    2954
  • Abstract
    The first mechanism-based inhibitor of a 3-deoxy-d-arabino heptulosonate 7-phosphate (DAH7P) synthase has been synthesised in 12 steps from d-arabinose, and has been found to be a very slow binding inhibitor of Escherichia coli DAH7P synthase.
  • Keywords
    DAHP , shikimate , DAH7P , Transition-state inhibitor
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2006
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    796904