• Title of article

    Peptoids as endothelin receptor antagonists

  • Author/Authors

    Falguni Dasgupta، نويسنده , , N. Gangadhar، نويسنده , , M. Bruhaspathy، نويسنده , , Ashwani K. Verma، نويسنده , , Simi Sarin، نويسنده , , Ashish K. Mukherjee، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2001
  • Pages
    3
  • From page
    555
  • To page
    557
  • Abstract
    A series of new peptoids as endothelin receptor antagonists has been synthesized. Screening them for their ability to bind with endothelin receptors (ETA and ETB) competitively in the presence of (125I) endothelin led to the discovery of compounds as possible leads with IC50s in the low micromolar concentrations.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2001
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    800394

    • Link To Document
    https://search.isc.ac/dl/search/defaultta.aspx?DTC=10&DC=800394