Author/Authors :
Guirong Qu، نويسنده , , Peng-Yang Xin، نويسنده , , Hong-Ying Niu، نويسنده , , Xin Jin، نويسنده , , Xiao-Ting Guo، نويسنده , , Xi-Ning Yang، نويسنده , , Hai-Ming Guo، نويسنده ,
Abstract :
An efficient method for the synthesis of 6-arylpurines (nucleosides) was developed via Suzuki–Miyaura cross-coupling reactions of 6-chloropurines (nucleosides) and sodium tetraarylborate in neat water (ethanol). The process gave good to high isolated yields within a short reaction time under microwave irradiated conditions.
Keywords :
palladium-catalyzed , Suzuki–Miyaura coupling , 6-Chloropurines , Sodium tetraarylborate , Water , Microwave-assisted synthesis