• Title of article

    A 3,4-Epoxypiperidine structure as a novel and simple DNA-cleavage unit

  • Author/Authors

    Kazuyuki Miyashita، نويسنده , , Myunji Park، نويسنده , , Sayako Adachi، نويسنده , , Sayori Seki، نويسنده , , Satoshi Obika، نويسنده , , Takeshi Imanishi، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2002
  • Pages
    3
  • From page
    1075
  • To page
    1077
  • Abstract
    Based on the 4-hydroxy-1-azabicyclo[3.1.0]hexane structure of azinomycin, a 3,4-epoxypiperidine structure was designed as a novel and simple alkylating molecular unit, and some 3,4-epoxypiperidine derivatives were found to show DNA-cleavage activity, the structural requirements for which were revealed.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2002
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    792143