• Title of article

    Liver X receptor antagonists with a phthalimide skeleton derived from thalidomide-related glucosidase inhibitors

  • Author/Authors

    Tomomi Noguchi-Yachide، نويسنده , , Atsushi Aoyama، نويسنده , , Makoto Makishima، نويسنده , , Hiroyuki Miyachi، نويسنده , , Yuichi Hashimoto، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2007
  • Pages
    5
  • From page
    3957
  • To page
    3961
  • Abstract
    α-Glucosidase inhibitors with a chlorinated phthalimide or a thiophthalimide skeleton, derived from thalidomide, were found to possess liver X receptor (LXR) antagonistic activity. Novel LXR antagonists with a 2′-substituted phenylphthalimide skeleton were obtained by structural development of glucosidase inhibitors derived from thalidomide.
  • Keywords
    Phthalimide , thalidomide , Liver X receptor (LXR) , Glucosidase , Antagonist
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2007
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    798347